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ISIS 3521 A synthetic phosphorothioate oligodeoxynucleotide. As an antisense molecule, ISIS 3521 hybridizes to the 3-untranslated region of the human protein kinase C (PKC-alpha) mRNA, thereby inhibiting PKC-alpha expression and growth of PKC-alpha-dependent tumor cells. Check for active clinical trials or closed clinical trials using this agent. (NCI Thesaurus)
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Synonym: | ![](https://webarchive.library.unt.edu/eot2008/20090511122123im_/http://www.cancer.gov/images/spacer.gif) | DNA, d(P-thio)(GTTCTCGCTGGTGAGTTTCA) | | ![](https://webarchive.library.unt.edu/eot2008/20090511122123im_/http://www.cancer.gov/images/spacer.gif) | US brand names: | ![](https://webarchive.library.unt.edu/eot2008/20090511122123im_/http://www.cancer.gov/images/spacer.gif) | Affinitac Affinitak | | ![](https://webarchive.library.unt.edu/eot2008/20090511122123im_/http://www.cancer.gov/images/spacer.gif) | Code names: | ![](https://webarchive.library.unt.edu/eot2008/20090511122123im_/http://www.cancer.gov/images/spacer.gif) | CGP 64128A LY900003 | | ![](https://webarchive.library.unt.edu/eot2008/20090511122123im_/http://www.cancer.gov/images/spacer.gif) |
Previous: | iron sucrose injection, IRX-2, Iscar, Iscomatrix, ISIS 2503 | Next: | ISIS 5132, isoniazid, isosulfan blue, isotretinoin, Isovorin |
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