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The Practice of Medicinal Chemistry
(Third Edition)
Copyright © 2008 Elsevier Ltd. All rights reserved
Edited by:
Camille Georges Wermuth
ISBN: 978-0-12-374194-3
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Table of Contents
Biography
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Pages xxv-xxvi
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Contributors
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Pages xxix-xxxiii
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Preface to the First Edition
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Pages xxxv-xxxvi
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Preface to the Second Edition
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Pages xxxvii-xxxviii
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Preface to the Third Edition
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Page xxxix
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Part I: General Aspects of Medicinal Chemistry
Part II: Lead Compound Discovery Strategies
Part III: Primary Exploration of Structure–Activity Relationships
Part IV: Substituents and Functions: Qualitative and Quantitative Aspects of Structure–Activity Relationships
Part V: Spatial Organization, Receptor Mapping and Molecular Modeling
Part VI: Chemical Modifications Infl uencing the Pharmacokinetic Properties
Part VII: Pharmaceutical and Chemical Means to Solubility and Formulation Problems
Part VIII: Development of New Drugs: Legal and Economic Aspects
Index
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Pages 923-942
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